HomeClinical StudyHistamine Receptors, Location-Agonist-Antagonist

Histamine Receptors, Location-Agonist-Antagonist

Histamine Receptors, Location-Agonist-Antagonist

HSTAMINE RECEPTORS  
Receptor Location Agonists Antagonists
H
1
Smooth muscle,
endothelium,
brain
Histaprodifen Mepyramine,
Loratadine
H
2
Gastric mucosa,
cardiac muscle,
mast cells, brain
Amthamine Ranitidine,
Tiotidine
H
3
Presynaptic
Brain, Myenteric
plexus, other
neurons
R-a-Methyl
histamine,
Imetit,
Immepip
Thioperamide,
Iodophenpro
pit
H4 Eosinophils,
neutrophils, CD4
T cells
Clobenpropit,
Imetit,
Clozapine
Thioperamide
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